CGP 36216 is a selective antagonist of GABAB receptors (IC50 = 43 ?M).{28184,28183} Its action is reversed by the GABAB receptor agonist baclofen.{28183} It is active at presynaptic, but not postsynaptic, receptors.{28183}
产品描述
A selective antagonist of GABAB receptors (IC50 = 43 ?M); active at presynaptic, but not postsynaptic, receptors
